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Search Results for " mchr1 (gpr24) "

4

Compounds

Cat No. Product Name Synonyms Targets
T11966 MCHR1 antagonist 2 HER , Melanin-concentrating Hormone Receptor (MCHR)
MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.
TP1996 MCH(human, mouse, rat) MCH (human, mouse, rat) GPR , Melanin-concentrating Hormone Receptor (MCHR)
MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors (IC50 values are 0.3 and 1.5 nM and EC50 values are 3.9 and 0.1 nM at MCH1 and MCH2 receptors respectively). Increase...
T8004 SNAP 94847 hydrochloride GPR , Melanin-concentrating Hormone Receptor (MCHR)
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
T5406 SNAP 94847 SNAP-94847 GPR , Melanin-concentrating Hormone Receptor (MCHR)
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM). It has anxiolytic and antidepressant activity and reduces food intake in mice.
TargetMol